| 產(chǎn)品編號(hào) | D58240 |
| 英文名稱 | Calmidazolium chloride |
| 中文名稱 | 鈣調(diào)蛋白抑制劑 |
| 別 名 | R 24571 |
| 克 隆 號(hào) | |
| CAS | 57265-65-3 |
| 理論分子量 | 687.7 kDa |
| 檢測(cè)分子量 | |
| 保存條件 | Powder: -20℃ for 3 years | In solvent: -80℃ for 1 year |
| 注意事項(xiàng) | This product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications. |
| 產(chǎn)品介紹 |
Calmidazolium chloride is a calmodulin (CaMK) antagonist (Kd = 3 nM), antagonizing CaM-dependent phosphodiesterase(IC50 = 0.15 μM) and calmodulin-induced activation of erythrocyte Ca2+-transporting ATPase(IC50 = 0.35 μM). Calmidazolium chloride also induces apoptosis in certain cancer cell lines. |